biomedicina slovenica


"BUTYRYLCHOLINESTERASE" : 63

  1. Maraković Nikola; Knežević Anamarija; Rončević Igor; Brazzolotto Xavier; Šinko Goran
    Enantioseparation, in vitro testing, and structural characterization of triple-binding reactivators of organophosphate-inhibited cholinesterases
    2020
  2. Zandona Antonio; Lihtar Gabriela; Maraković Nikola; Miš Katarina; Bušić Valentina; Gašo-Sokač Dajana; Pirkmajer Sergej; Katalinić Maja
    Vitamin B3-based biologically active compounds as inhibitors of human cholinesterases
    2020
  3. Knez Damijan; Sosič Izidor; Mitrović Ana; Pišlar Anja; Kos Janko; Gobec Stanislav
    8-hydroxyquinoline-based anti-Alzheimer multimodal agents
    2020
  4. Pajk Stane; Knez Damijan; Košak Urban; Zorović Maja; Brazzolotto Xavier; Coquelle Nicolas; Nachon Florian; Colletier Jacques-Philippe; Živin Marko; Stojan Jure; Gobec Stanislav
    Development of potent reversible selective inhibitors of butyrylcholinesterase as fluorescent probes
    2020
  5. Mukhametgalieva Aliya R.; Aglyamova Aliya R.; Lushchekina Sofya V.; Goličnik Marko; Masson Patrick
    Time course of human cholinesterases-catalyzed competing substrate kinetics
    2019
  6. Stojan Jure
    The mechanism and benefit of human butyrylcholinesterase activation by what would otherwise be inhibitors
    2019
  7. Stojan Jure
    Rapid mechanistic evaluation and parameter estimation of putative inhibitors in a single-step progress-curve analysis
    2017
  8. Zorbaz Tamara; Braïki Anissa; Maraković Nikola; Renou Julien; Mora Eugenio; Maček Hrvat Nikolina; Katalinić Maja; Silman Israel; Sussman Joel; Mercey Guillaume
    Potent 3-hydroxy-2-pyridine aldoxime reactivators of organophosphate-inhibited cholinesterases with predicted blood-brain barrier penetration
    2018
  9. Maraković Nikola; Knežević Anamarija; Vinković Vladimir; Kovarik Zrinka; Šinko Goran
    Design and synthesis of N-substituted-2-hydroxyiminoacetamides and interactions with cholinesterases
    2016
  10. Bosak Anita; Knežević Anamarija; Gazić Smilović Ivana; Šinko Goran; Kovarik Zrinka
    Resorcinol-, catechol- and saligenin-based bronchodilating [beta]2-agonists as inhibitors of human cholinesterase activity
    2017
  11. Bosak Anita; Ramić Alma; Šmidlehner Tamara; Hrenar Tomica; Primožič Ines; Kovarik Zrinka
    Design and evaluation of selective butyrylcholinesterase inhibitors based on Cinchona alkaloid scaffold
    2018
  12. Knez Damijan; Coquelle Nicolas; Pišlar Anja; Žakelj Simon; Jukič Marko; Sova Matej; Mravljak Janez; Nachon Florian; Brazzolotto Xavier; Kos Janko; Colletier Jacques-Philippe; Gobec Stanislav
    Multi-target-directed ligands for treating Alzheimer's disease
    2018
  13. Brvar Miran; Chan Ming Yin; Dawson Andrew H.; Ribchester Richard R.; Eddleston Michael
    Magnesium sulfate and calcium channel blocking drugs as antidotes for acute organophosphorus insecticide poisoning - a systematic review and meta-analysis
    2018
  14. Panek Dawid; Więckowska Anna; Pasieka Anna; Godyń Justyna; Jończyk Jakub; Bajda Marek; Knez Damijan; Gobec Stanislav; Malawska Barbara
    Design, synthesis, and biological evaluation of 2-(benzylamino-2-hydroxyalkyl)isoindoline-1,3-diones derivatives as potential disease-modifying multifunctional anti-Alzheimer agents
    2018
  15. Košak Urban; Brus Boris; Knez Damijan; Žakelj Simon; Trontelj Jurij; Pišlar Anja; Šink Roman; Jukič Marko; Živin Marko; Podkowa Adrian; Nachon Florian; Brazzolotto Xavier; Stojan Jure; Kos Janko; Coquelle Nicolas; Sałat Kinga; Colletier Jacques-Philippe; Gobec Stanislav
    The magic of crystal structure-based Inhibitor optimization
    2018
  16. Šinko Goran; Maraković Nikola; Stojan Jure
    Evaluation of butyrylcholinesterase stereoselectivity in interaction with enantiomers of ethopropazine
    2014
  17. Stojan Jure
    The significance of low substrate concentration measurements for mechanistic interpretation in cholinesterases
    2013
  18. Bartolucci Cecilia; Stojan Jure; Yu Qian-Sheng; Greig Nigel H; Lamba Doriano
    Kinetics of Torpedo californica acetylcholinesterase inhibition by bisnorcymserine and crystal structure of the complex with its leaving group
    2012
  19. Šinko Goran; Kovarik Zrinka; Reiner Elsa; Simeon-Rudolf Vera; Stojan Jure
    Mechanism of stereoselective interaction between butyrylcholinesterase and ethopropazine enantiomers
    2011
  20. Fekonja Ota; Zorec-Karlovšek Majda; El Kharbili Manale; Fournier Didier; Stojan Jure
    Inhibition and protection of cholinesterases by methanol and ethanol
    2007
  21. Frasco Manuela F; Colletier Jacques-Philippe; Weik Martin; Carvalho Félix; Guilhermino Lúcia; Stojan Jure; Fournier Didier
    Mechanisms of cholinesterase inhibition by inorganic mercury
    2007
  22. Šinko Goran; Stojan Jure; Goličnik Marko; Grubič Zoran; Kovarik Zrinka; Simeon-Rudolf Vera
    Butyrylcholinesterase inhibition by ethopropazine enantiomers: evaluation of kinetic models
    2006
  23. Miš Katarina
    Colocalization of acetylcholinesterase, butyrylcholinesterase and choline acetyltransferase in rat spinal cord
    2005
  24. Brvar Miran; Možina Martin; Bunc Matjaž
    Poisoning with rivastigmine
    2005
  25. Miš Katarina
    Izražanje živčnomišičnih komponent v hrbtenjači sesalca
    [Expression of the neuromuscular components in the mammalian spinal cord]
    2004
  26. Reiner Elsa; Šinko Goran; Bosak Anita; Simeon-Rudolf Vera; Radić Zoran; Taylor Palmer; Stojan Jure; Goličnik Marko
    Kinetics of ethopropazine binding to butyrylcholinesterase in the absence and presence of acetylthiocholine
    2004
  27. Simeon-Rudolf Vera; Šinko Goran; Štuglin Anita; Stojan Jure; Goličnik Marko; Reiner Elsa
    Comparison of two reaction schemes for the hydrolysis of acetylthiocholine by butyrylcholinesterase
    2004
  28. Reiner Elsa; Šinko Goran; Štuglin Anita; Simeon-Rudolf Vera; Radić Goran; Taylor Palmer; Stojan Jure; Goličnik Marko
    Kinetics of ethopropazine binding to butyrylcholinesterase in the absence and presence of acetylthiocholine
    2002
  29. Miš Katarina; Marš Tomaž; Jevšek Marko; Brank Martina; Zajc-Kreft Katarina; Grubič Zoran
    Localization of mRNAs encoding acetylcholinesterase and butyrylcholinesterase in the rat spinal cord by nonradioactive in situ hybdrization
    2003
  30. Miš Katarina; Davidson Edgar; Park Hyejeong; King Michael P; Marš Tomaž; Jevšek Marko; Brank Martina; Grubić Zoran
    mRNAs encording acteylcholinesterase, butyrylcholinesterase, and agrin 19, share the same temporal pattern of expression during development of rat spinal cord
    2004
  31. Kogoj Aleš
    Vloga butirilholinesteraze pri zdravljenju Alzheimerjeve bolezni
    2002
  32. Goličnik Marko
    Mehanizem kooperativnih pojavov pri holinesterazah
    [Mechanism of cooperative phenomena by cholinesterases]
    2002
  33. Goličnik Marko; Stojan Jure
    Multi-step analysis as a tool for kinetic parameter estimation and mechanism discrimination in the reaction between tight-binding fasciculin 2 and electric eel acetylcholinesterase
    2002
  34. Simeon-Rudolf Vera; Sinko Goran; Stuglin Anita; Stojan Jure; Goličnik Marko; Reiner Elsa
    Comparison of two reaction schemes for the hydrolysis of acetylcholine by butyrylcholinesterase
    2002
  35. Stojan Jure; Goličnik Marko; Froment Marie-Therese; Estour Francois; Masson Patrick
    Concentration-dependent reversible activation-inhibition of human butyrylcholinesterase by tetraethylammonium ion
    2002
  36. Goličnik Marko; Šinko Goran; Simeon-Rudolf Vera; Grubič Zoran; Stojan Jure
    Kinetic model of ethopropazine interaction with horse serum butyrylcholinesterase and its docking into the active site
    2002
  37. Murko-Bulić Jožica; Miš Katarina; Davidson Edgar; Park Hyejeong; King Michael P; Marš Tomaž; Grubič Zoran
    Expression of butyrylcholinesterase mRNA in rat spinal cord
    2001
  38. Weber Urša
    Vpliv glukokortikoidov na ekspresijo acetilholinesterase in butirilholinesterase v možganih in jetrih sesalca
    [Glucocorticoid influence on acetylcholinesterase and butyrylcholinesterase expression in mammalian brain and liver]
    1998
  39. Masson Patrick; Nachon Florian; Xie Weihua; Froment Marie-Therese; Weingand-Ziade Alexandra; Goeldner Maurice; Lockridge Oksana
    The peripheral anionic site of butyrylcholinesterase: from facts to functions
    [Periferno anionsko mesto na butilholinesterazi: od dejstev k vlogi]
    2000
  40. Pavlič MR; Zorko M
    The role of water of hydration in acylation of butyrylcholinesterase
    1985
  41. Brzin M
    Biological functions of acetylcholinesterase and butyrylcholinesterase, and changes in disease states. Introduction
    1984
  42. Pavlin R
    Activity of total cholinesterase, butyrylcholinesterase, tyrosine hydroxylase, dopa- and glutamic acid decarboxylase within single nerve cells isolated form substantia nigra and reticular formation of man and rat
    1983
  43. Pavlič MR; Zorko M
    THE ROLE OF WATER OF HYDRATION IN ACYLATION OF BUTYRYLCHOLINESTERASE
    1982
  44. Pavlič MR
    THE ACCELERATION OF METHANESULFONYLATION OF BUTYRYLCHOLINESTERASE WITH CATIONIC ACCELERATORS
    1981
  45. Goličnik Marko; Masson Patrick; Stojan Jure
    Two time periods of acetylthiocholine hydrolysis by human W82A butyrylcholinesterase
    2000
  46. Simeon-Rudolf Vera; Reiner Elsa; Šinko Goran; Štuglin Anita; Goličnik Marko; Stojan Jure
    Competitive and non-competitive inhibition of horse serum butyrylcholinesterase by ethopropazine
    2000
  47. Stojan Jure; Sinko Goran; Goličnik Marko; Simeon-Rudolf Vera; Reiner Elsa
    Interaction of wild type horse serum butyrylcholinesterase with ethopropazine
    2000
  48. Simeon-Rudolf Vera; Evans Robert T
    Interlaboratory study of the proficiency of butyrylcholinesterase activity measurements
    1999
  49. Simeon-Rudolf Vera; Šinko Goran; Reiner Elsa
    Inhibition of human serum butyrylcholinesterase phenotypes by ethopropazine
    1999
  50. Estour Francois; Stojan Jure; Froment Marie-Therese; Masson Patrick
    Mechanism of activation and inhibition of butyrylcholinesterase by tetraalkylammonium salts
    1999
  51. Masson Patrick; Nachon Florian; Xie Wue Hua; Froment Marie-Therese; Weingand-Ziade Alexandra; Goeldner Maurice; Lockridge Oksana
    The peripheral anionic site of butyrylcholinesterase: from facts to functions
    1999
  52. Weber Urška; Brank Martina; Grubič Zoran
    Glucocorticoids differentially control synthesis of acetylcholinesterase and butyrylcholinesterase in rat liver and brain
    1999
  53. Stojan Jure; Marcel Veronique; Estrada-Mondaca Sandino; Klaebe Alain; Masson Patrick; Fournier Didier
    A putative kinetic model for substrate metabolisation by Drosophila acetylcholinesterase
    1998
  54. Sepčić Kristina; Turk Tom; Maček Peter
    Anticholinesterase activity of the fluorescent zoanthid pigment, parazoanthoxanthin A
    1998
  55. Weber U; Brank M; Grubič Z
    Glucocorticoids differentially control synthesis of acetylcholinesterase and butyrylcholinesterase in rat liver and brain
    1998
  56. Quinn Daniel M.
    Enzymes of the cholinesterase family. 5th international Meeting on Cholinesterases September 24-28, 1994, Madras, India
    1995
  57. Stojan Jure; Pavlič Miloš R
    Mechanism of eserine action on the hydrolysis of butyrylthiocholine by butyrylcholinesterase
    1997
  58. Novak-Antolič Ž
    Študij mediatorskih sistemov v humanem miometriju
    1989
  59. Alif M
    Termična denaturacija butirilholinesteraze
    1989
  60. Grubič Z; Sket D; Brzin M
    Iso-OMPA-induced potentiation of soman toxicity in rat correlates with the inhibition of plasma carboxylesterases
    1988
  61. Sepp A; Palumaa P; Langel U; Jaerv J; Zorko M
    Spatial orientation of n-alkanesulfonyl chlorides in the active center of cholinesterases
    1989
  62. Gadžijev E
    Regeneracijska sposobnost podganjih jeter po obsežni resekciji: vpliv anabolnih hormonov
    1988
  63. Zorko M; Stojan J; Pavlič MR
    Influence of ionic strength on the interaction between D-tubocurarine and cholinesterases
    1986


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